1) "Principles of Biochemistry" 4th edition by Horton et al., Pearson Education, ISBN:9780131977365
2) "Organic Chemistry - A biological approach" 2nd edition by John McMurry, Thomson Brooks/Cole, Cengage learning, ISBN: 9780495391470 (if you have the first edition, this is also fine)
3) Additional material will be made available free of charge during the course (e.g. concerning the drug design part of the course).